SCHEMBL11405171

SCHEMBL11405171

O=C1CCC(c2ccc(-c3ccc(F)cc3)cc2)=NN1c1ccncc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.53
CA12 O43570 3/20 0.47
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
CA9 Q16790 3/20 0.47
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
MAPK14 Q16539 2/20 0.44
MT-CO2 P00403 1/20 0.41
PTGS1 P23219 2/20 0.39
PTGS2 P35354 2/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29395562 0.85 PDE4A (0.60) GAACA12CA1CA2CA9
SCHEMBL11397866 0.84 MAPT (0.49) GAACA12CA1CA2CA9
SCHEMBL23534153 0.81 GAA (0.54) GAACA12CA1CA2CA9
SCHEMBL29394932 0.77 CA12 (0.68) GAACA12CA1CA2CA9
SCHEMBL11398931 0.77 CD274 (0.59) GAACA12CA1CA2CA9
SCHEMBL11399660 0.74 PDE4B (0.55) GAAPDE4APDE4BPDE4CPDE4D
SCHEMBL6014889 0.73 CA12 (0.71) GAACA12CA1CA2CA9
SCHEMBL29394845 0.73 PDE4A (0.56) GAACA12CA1CA2CA9
SCHEMBL21144550 0.72 PDE4B (0.52) GAAPDE4APDE4BPDE4CPDE4D
SCHEMBL11732162 0.72 MEN1 (0.61) GAACA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4289774-A Lipid lowering and anti-thrombotic 6-arylpyridazin-3-ones and a process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-09-15 US disclosed
EP-0010156-A1 6-Arylpyridazine-3-ones, pharmaceutical compositions containing them and process for their preparation MERCK PATENT GmbH (DE) 1980-04-30 EP disclosed