SCHEMBL1147788

SCHEMBL1147788

COc1ccc2nccc(CCC3(O)CCC(C(=O)Nc4ccc(C)c(F)c4)CC3)c2n1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.45
TP53 P04637 1/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 1/20 0.40
SLC2A1 P11166 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3250867 0.87 KCNH2 (0.43) KCNH2SLC2A1
SCHEMBL1148084 0.86 KCNH2 (0.41) KCNH2
SCHEMBL1147476 0.86 KCNH2 (0.52) KCNH2KDM4ESMN1; SMN2MAPT
SCHEMBL1147947 0.86 KCNH2 (0.52) KCNH2KDM4ESMN1; SMN2MAPT
SCHEMBL1147907 0.83 TRPV1 (0.43) KCNH2
SCHEMBL1147704 0.83 TRPV1 (0.43) KCNH2
SCHEMBL3251999 0.81 KCNH2 (0.44) KCNH2
SCHEMBL3243307 0.81 KCNH2 (0.44) KCNH2
SCHEMBL3251995 0.81 KCNH2 (0.44) KCNH2
SCHEMBL1147900 0.80 KCNH2 (0.42) KCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7888359-B2 Cyclohexyl or piperidinyl carboxamide antibiotic derivatives ACTELION PHARMACEUTICAL LTD. (CH) 2011-02-15 US claimed
US-7888359-B2 Cyclohexyl or piperidinyl carboxamide antibiotic derivatives ACTELION PHARMACEUTICAL LTD. (CH) 2011-02-15 US disclosed