SCHEMBL11540642

SCHEMBL11540642

CC(CCl)c1ccc(-c2ccc(F)cc2F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 4/20 0.41
CYP2C9 P11712 3/20 0.41
APP P05067 3/20 0.41
CYP3A4 P08684 3/20 0.41
GRM2 Q14416 2/20 0.41
HTR2A P28223 1/20 0.41
AKR1C3 P42330 4/20 0.41
AKR1C2 P52895 4/20 0.41
PTGS1 P23219 3/20 0.41
MEN1 O00255 2/20 0.41
PTGS2 P35354 2/20 0.41
KMT2A Q03164 2/20 0.41
PSEN1 P49768 2/20 0.41
PSEN2 P49810 2/20 0.41
APH1B Q8WW43 2/20 0.41
NCSTN Q92542 2/20 0.41
APH1A Q96BI3 2/20 0.41
PSENEN Q9NZ42 2/20 0.41
FABP2 P12104 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11543436 0.85 CYP2C19 (0.46) CYP2C19CYP2C9APPCYP3A4AKR1C3
SCHEMBL11542595 0.84 CYP2C19 (0.41) CYP2C19CYP2C9APPCYP3A4GRM2
SCHEMBL11545076 0.83 AKR1C3 (0.45) CYP2C19CYP2C9APPCYP3A4AKR1C3
SCHEMBL11544423 0.83 CYP2C19 (0.43) CYP2C19CYP2C9APPCYP3A4GRM2
SCHEMBL11622662 0.81 APP (0.44) CYP2C19CYP2C9APPCYP3A4GRM2
SCHEMBL11543758 0.81 AKR1C3 (0.41) CYP2C19CYP2C9APPCYP3A4GRM2
SCHEMBL12418419 0.81 APP (0.46) CYP2C19CYP2C9APPCYP3A4AKR1C3
SCHEMBL11542959 0.81 APP (0.46) CYP2C19CYP2C9APPCYP3A4AKR1C3
SCHEMBL11545400 0.80 CYP2C19 (0.40) CYP2C19CYP2C9APPCYP3A4GRM2
SCHEMBL11542929 0.79 FFAR1 (0.51) CYP2C19CYP2C9APPCYP3A4AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4151302-A Araliphatic dihalogen compounds composition and method of use MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-04-24 US disclosed
US-4057647-A Araliphatic dihalogen compounds and process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-11-08 US disclosed