SCHEMBL11540905

SCHEMBL11540905

COc1cc2c(c(C(N)=O)c1OC)CCNCC2c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 18/20 0.53
DRD5 P21918 4/20 0.53
DRD2 P14416 8/20 0.49
KDM4E B2RXH2 5/20 0.49
MAPT P10636 3/20 0.49
CYP3A4 P08684 2/20 0.49
NFKB1 P19838 2/20 0.49
THPO P40225 2/20 0.49
HIF1A Q16665 2/20 0.49
HSD17B10 Q99714 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
PKM P14618 1/20 0.49
RECQL P46063 1/20 0.49
MTOR P42345 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MAPK1 P28482 2/20 0.48
BLM P54132 2/20 0.48
GFER P55789 2/20 0.48
GALR3 O60755 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11245963 0.90 DRD1 (0.54) DRD1DRD5DRD2KDM4EMAPT
SCHEMBL11539154 0.89 DRD1 (0.53) DRD1DRD5DRD2KDM4EMAPT
Hydrochloric Acid SCHEMBL11267852 0.89 DRD1 (0.53) DRD1DRD5DRD2KDM4EMAPT
SCHEMBL14494976 0.84 DRD1 (0.58) DRD1DRD5DRD2KDM4EMAPT
Hydrochloric Acid SCHEMBL11262498 0.82 DRD1 (0.44) DRD1DRD5DRD2KDM4EMAPT
Hydrochloric Acid SCHEMBL11253551 0.82 DRD1 (0.56) DRD1DRD5DRD2KDM4EMAPT
Hydrochloric Acid SCHEMBL11539700 0.82 DRD1 (0.46) DRD1DRD5DRD2KDM4EMAPT
SCHEMBL7329076 0.81 DRD1 (0.55) DRD1DRD5DRD2KDM4EMAPT
SCHEMBL7331849 0.81 DRD1 (0.60) DRD1DRD5DRD2KDM4EMAPT
SCHEMBL11265194 0.81 DRD1 (0.55) DRD1DRD5DRD2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4165372-A 6-Carboxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine compounds and use as dopaminergic agents SMITHKLINE CORPORATION (US) 1979-08-21 US disclosed