SCHEMBL11545101

SCHEMBL11545101

NC(=O)c1cn[c]nc1-c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.42
TGFBR1 P36897 2/20 0.42
TGFBR2 P37173 1/20 0.42
PARP1 P09874 2/20 0.40
CYP2A6 P11509 1/20 0.39
DHODH Q02127 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
CDC7 O00311 1/20 0.39
CHEK2 O96017 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
KDM4E B2RXH2 3/20 0.37
P4HTM Q9NXG6 2/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
METAP1 P53582 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3620548 0.78 GRM5 (0.51) GRM5TGFBR1TGFBR2PARP1DHODH
SCHEMBL11576372 0.77 HPGD (0.45) LMNACYP1A2POLBALDH1A1HPGD
SCHEMBL29455925 0.76 GRM5 (0.50) GRM5TGFBR1TGFBR2PARP1DHODH
SCHEMBL11546311 0.76 KDM4E (0.43) CYP2A6KDM4EP4HTMLMNACYP1A2
SCHEMBL20985616 0.74 KDM4E (0.45) TGFBR1CYP2A6KDM4EP4HTMLMNA
SCHEMBL22584044 0.73 NPSR1 (0.46) GRM5TGFBR1TGFBR2PARP1DHODH
SCHEMBL558611 0.73 KDM4E (0.43) CYP2A6KDM4EP4HTMLMNACYP1A2
Dipyridyl SCHEMBL20448088 0.71 KDM4E (0.67) PARP1CYP2A6KDM4EP4HTMLMNA
SCHEMBL19581487 0.71 GRM5 (0.45) GRM5TGFBR1TGFBR2PARP1DHODH
SCHEMBL2943452 0.71 GRM5 (0.54) GRM5PARP1DHODHPARP2CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed