SCHEMBL11552121

SCHEMBL11552121

CCOc1ccc(C(=O)c2c(-c3ccc(OC)cc3)sc3cc(O)ccc23)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 18/20 0.69
ESR2 Q92731 9/20 0.69
CNR1 P21554 2/20 0.62
CNR2 P34972 1/20 0.62
MEN1 O00255 1/20 0.60
PLD2 O14939 1/20 0.60
KDM1A O60341 1/20 0.60
NR1I2 O75469 1/20 0.60
USP2 O75604 1/20 0.60
ALDH1A1 P00352 1/20 0.60
C5 P01031 1/20 0.60
LMNA P02545 1/20 0.60
TP53 P04637 1/20 0.60
FYN P06241 1/20 0.60
PGR P06401 1/20 0.60
CYP3A4 P08684 1/20 0.60
ADRA2A P08913 1/20 0.60
ADORA3 P0DMS8 1/20 0.60
CYP2D6 P10635 1/20 0.60
MAPT P10636 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30558217 0.94 ESR1 (0.70) ESR1ESR2CNR1MEN1PLD2
SCHEMBL11546753 0.93 ESR1 (0.69) ESR1ESR2CNR1CNR2MEN1
SCHEMBL6425122 0.92 ESR1 (0.68) ESR1ESR2CNR1CNR2TDP1
SCHEMBL7075381 0.92 ESR1 (0.72) ESR1ESR2CNR1CNR2MEN1
SCHEMBL7075631 0.91 ESR1 (0.74) ESR1ESR2CNR1CNR2MEN1
SCHEMBL7075664 0.91 ESR1 (0.74) ESR1ESR2CNR1CNR2MEN1
SCHEMBL11546633 0.90 ESR1 (0.67) ESR1ESR2CNR1MEN1PLD2
SCHEMBL11550082 0.90 ESR1 (0.63) ESR1ESR2CNR1MEN1PLD2
SCHEMBL7971665 0.88 ESR1 (0.66) ESR1ESR2CNR1MEN1PLD2
SCHEMBL11551310 0.86 ESR1 (0.65) ESR1ESR2CNR1CNR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4133814-A ANTITUMOR AGENTS ELI LILLY AND COMPANY (US) 1979-01-09 US disclosed