SCHEMBL11567653

SCHEMBL11567653

CN(C)C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.69
APEX1 P27695 1/20 0.67
PDK1 Q15118 1/20 0.62
TRPV1 Q8NER1 2/20 0.58
TP53 P04637 1/20 0.56
SLC6A3 Q01959 1/20 0.56
GRM4 Q14833 1/20 0.56
LMNA P02545 2/20 0.55
RAF1 P04049 1/20 0.55
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA7 P43166 1/20 0.54
CA9 Q16790 1/20 0.54
MEN1 O00255 1/20 0.54
HTT P42858 1/20 0.54
KMT2A Q03164 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
TMPRSS4 Q9NRS4 1/20 0.54
KCNJ5 P48544 1/20 0.54
KCNJ3 P48549 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11632558 0.90 KDR (0.68) KDRAPEX1PDK1TRPV1SLC6A3
SCHEMBL11201462 0.88 APEX1 (0.67) KDRAPEX1PDK1TRPV1TP53
SCHEMBL10222082 0.84 KDR (0.59) KDRAPEX1PDK1TRPV1SLC6A3
SCHEMBL10913149 0.83 TP53 (0.57) KDRAPEX1TRPV1TP53CA1
SCHEMBL462753 0.83 KDR (0.76) KDRPDK1TRPV1GRM4LMNA
SCHEMBL16628095 0.83 TRPV1 (0.65) KDRPDK1TRPV1SLC6A3GRM4
SCHEMBL11092519 0.82 RAF1 (0.59) TP53LMNARAF1CA1CA2
SCHEMBL118026 0.82 KDR (1.00) KDRPDK1TRPV1GRM4CA1
SCHEMBL29364392 0.82 KDR (1.00) KDRPDK1TRPV1GRM4CA1
SCHEMBL848037 0.82 MAPT (0.60) APEX1TP53LMNARAF1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4137068-A Novel ureas ROUSSEL UCLAF (FR) 1979-01-30 US disclosed
US-3931311-A N,N,N-trisubstituted N-halogenomethylurea and thiourea compounds and process for their preparation BAYER AKTIENGESELLSCHAFT (DT) 1976-01-06 US disclosed