SCHEMBL11577101

SCHEMBL11577101

CN1CCC(C2(O)c3ccc(Cl)cc3Oc3ccc(F)cc32)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.43
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAP3K14 Q99558 1/20 0.38
DRD2 P14416 6/20 0.35
DRD4 P21917 6/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C19 P33261 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HTR2C P28335 3/20 0.34
HTR2B P41595 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RAD52 P43351 2/20 0.34
HTR2A P28223 3/20 0.34
CHRM2 P08172 2/20 0.34
HTR1A P08908 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11574266 0.86 MAPK1 (0.54) HRH4MAPK1SMN1; SMN2DRD2DRD4
SCHEMBL11575421 0.84 SMN1; SMN2 (0.54) HRH4MAPK1SMN1; SMN2DRD2DRD4
SCHEMBL11574683 0.78 RAD52 (0.47) HRH4MAPK1SMN1; SMN2DRD2DRD4
SCHEMBL11574348 0.75 MAPK1 (0.59) MAPK1SMN1; SMN2MAP3K14DRD2DRD4
SCHEMBL11573321 0.72 MAPK1 (0.54) MAPK1SMN1; SMN2DRD2DRD4HTR2B
SCHEMBL11574851 0.72 SMN1; SMN2 (0.54) MAPK1SMN1; SMN2DRD2DRD4CYP1A2
SCHEMBL11574443 0.71 MAPK1 (0.46) MAPK1SMN1; SMN2DRD2TP53MAPT
SCHEMBL11577080 0.70 SMN1; SMN2 (0.55) MAPK1SMN1; SMN2MAP3K14DRD2DRD4
SCHEMBL10409949 0.70 MAPK1 (0.79) MAPK1SMN1; SMN2DRD2HTR2BL3MBTL1
SCHEMBL11575959 0.70 MAPK1 (0.51) MAPK1SMN1; SMN2DRD2DRD4L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4086350-A FLUORO, CHLORO AND CYANO SUBSTITUTED 4-(9-XANTHENYLIDENE, 9-THIOXANTHENYLIDENE OR 11(6H)-DIBENZO(B,E)OXEPINYLIDENE)-1-METHYL-PIPERIDINES SMITHKLINE CORPORATION (US) 1978-04-25 US disclosed