SCHEMBL11599290

SCHEMBL11599290

FC(F)(F)c1ccc(C(Cl)(Cl)Cl)cc1Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.58
PDE2A O00408 3/20 0.49
CYP3A4 P08684 1/20 0.45
MAPK1 P28482 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CES2 O00748 2/20 0.38
NOTUM Q6P988 3/20 0.38
RAPGEF3 O95398 1/20 0.36
KMO O15229 2/20 0.36
DAO P14920 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.35
IDO1 P14902 1/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3A P46098 1/20 0.34
HTR3D Q70Z44 1/20 0.34
HTR3C Q8WXA8 1/20 0.34
KDR P35968 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3789260 0.86 PDE2A (0.56) TSHRPDE2ACES2KMODAO
SCHEMBL8425257 0.84 TSHR (0.65) TSHRPDE2ACYP3A4MAPK1TDP1
SCHEMBL5381489 0.83 TSHR (0.58) TSHRNOTUMIDO1HTR3EHTR3B
SCHEMBL11599763 0.83 PDE2A (0.57) TSHRPDE2ACYP3A4MAPK1TDP1
SCHEMBL4792259 0.81 PDE2A (0.51) PDE2ATDP1CES2NOTUMRAPGEF3
SCHEMBL11598716 0.78 PDE2A (0.53) TSHRPDE2ACYP3A4MAPK1TDP1
SCHEMBL11600948 0.78 TSHR (0.56) TSHRPDE2ACYP3A4MAPK1TDP1
SCHEMBL11600693 0.78 PDE2A (0.57) TSHRPDE2ACYP3A4MAPK1TDP1
SCHEMBL11598957 0.78 TSHR (0.56) TSHRPDE2ACYP3A4MAPK1TDP1
SCHEMBL29129641 0.76 PDE2A (0.41) TSHRPDE2ACES2NOTUMRAPGEF3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4079089-A CONTACTING A BIS/TRICHLOROMETHYL/-BENZENE WITH HYDROGEN FLUORIDE, HALOGEN TRANSFER CATALYST BAYER AKTIENGESELLSCHAFT (DT) 1978-03-14 US disclosed