SCHEMBL11599689

SCHEMBL11599689

O=C(c1ccccc1)c1sc2cc(O)ccc2c1-c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 15/20 0.71
CLK1 P49759 1/20 0.47
DYRK1A Q13627 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
ESR2 Q92731 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
USP2 O75604 1/20 0.43
GAA P10253 1/20 0.43
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8341396 0.96 ESR1 (0.76) ESR1CLK1DYRK1ADYRK1BESR2
SCHEMBL8338171 0.93 ESR1 (0.63) ESR1CLK1DYRK1ADYRK1B
SCHEMBL11600001 0.91 ESR1 (0.67) ESR1ESR2
SCHEMBL21260801 0.91 ESR1 (0.78) ESR1CLK1DYRK1ADYRK1BESR2
SCHEMBL11600909 0.89 ESR1 (0.58) ESR1ESR2
SCHEMBL11598721 0.89 ESR1 (0.56) ESR1CLK1DYRK1ADYRK1BMEN1
SCHEMBL21261046 0.88 ESR1 (0.63) ESR1CLK1DYRK1ADYRK1BESR2
SCHEMBL21260814 0.87 ESR1 (0.62) ESR1CLK1DYRK1ADYRK1BESR2
SCHEMBL21260850 0.87 ESR1 (0.62) ESR1CLK1DYRK1ADYRK1BESR2
SCHEMBL21260976 0.87 ESR1 (0.62) ESR1CLK1DYRK1ADYRK1BESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4075227-A NONSTEROIDAL ELI LILLY AND COMPANY (US) 1978-02-21 US disclosed