SCHEMBL11600683

SCHEMBL11600683

CCOc1ccc2c(-c3ccc(OCCN4CCCCC4)cc3)c(C(=O)c3ccccc3)sc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 17/20 0.60
ESR2 Q92731 17/20 0.60
ENPP3 O14638 1/20 0.56
MEN1 O00255 1/20 0.54
PLD2 O14939 1/20 0.54
KDM1A O60341 1/20 0.54
NR1I2 O75469 1/20 0.54
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
C5 P01031 1/20 0.54
LMNA P02545 1/20 0.54
TP53 P04637 1/20 0.54
FYN P06241 1/20 0.54
PGR P06401 1/20 0.54
CYP3A4 P08684 1/20 0.54
ADRA2A P08913 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CYP2D6 P10635 1/20 0.54
MAPT P10636 1/20 0.54
CYP2C9 P11712 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11599867 0.93 ESR1 (0.70) ESR1ESR2ENPP3LTA4H
SCHEMBL11602492 0.88 ESR1 (0.59) ESR1ESR2LTA4H
SCHEMBL11551601 0.88 ESR1 (0.75) ESR1ESR2ENPP3MEN1PLD2
SCHEMBL20747941 0.86 ESR1 (0.68) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL11602238 0.86 ESR1 (0.76) ESR1ESR2ENPP3MEN1PLD2
SCHEMBL11598939 0.84 UBE2N (0.61) ESR1ESR2ENPP3ALDH1A1KDM4E
SCHEMBL11600046 0.83 ESR1 (0.58) ESR1ESR2
SCHEMBL11602415 0.83 ESR1 (0.67) ESR1ESR2MEN1PLD2KDM1A
SCHEMBL11601741 0.83 ESR1 (0.75) ESR1ESR2ENPP3LTA4H
SCHEMBL11209650 0.83 ESR1 (0.82) ESR1ESR2ENPP3MEN1PLD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4075227-A NONSTEROIDAL ELI LILLY AND COMPANY (US) 1978-02-21 US disclosed