SCHEMBL11603000

SCHEMBL11603000

Cn1cc(CCS)c2ccccc21

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.69
GPR84 Q9NQS5 1/20 0.67
KEAP1 Q14145 1/20 0.58
NFE2L2 Q16236 1/20 0.58
SLC6A4 P31645 1/20 0.52
CA2 P00918 1/20 0.50
KDM4E B2RXH2 1/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
ALDH1A1 P00352 2/20 0.49
IMPDH2 P12268 1/20 0.49
TP53 P04637 2/20 0.48
LMNA P02545 2/20 0.48
GLA P06280 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
AHR P35869 2/20 0.47
TSHR P16473 1/20 0.47
HTR6 P50406 1/20 0.46
RXFP1 Q9HBX9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7004405 0.85 HTR2A (0.73) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL9889542 0.83 HTR2A (0.71) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL12850609 0.82 HTR2A (0.65) HTR2AGPR84KEAP1NFE2L2HTR6
SCHEMBL9206509 0.81 HTR2A (0.69) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL7391194 0.81 HTR2A (0.69) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL11359977 0.81 HTR2A (0.69) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL5598636 0.81 HTR2A (0.69) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL18328036 0.81 HTR2A (0.69) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL5402680 0.81 HTR2A (0.69) HTR2AGPR84KEAP1NFE2L2SLC6A4
SCHEMBL332959 0.81 HTR2A (1.00) HTR2AGPR84KEAP1NFE2L2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4066780-A Pyranoindole derivatives as antiulcer agents AYERST MCKENNA AND HARRISON LTD. (CA) 1978-01-03 US disclosed
US-4066779-A ANTIDEPRESSANT, ANTIULCER AYERST, MCKENNA AND HARRISON LTD. (CA) 1978-01-03 US disclosed
US-4041169-A TREATING AND PREVENTING ULCERS AYERST MCKENNA AND HARRISON LTD. (CA) 1977-08-09 US disclosed
US-4003913-A ANTIDEPRESSANTS, ANTIULCER AGENTS AYERST MCKENNA AND HARRISON LTD. (CA) 1977-01-18 US disclosed