SCHEMBL11623975

SCHEMBL11623975

Cc1cccc(-c2ccc3nnc(C)n3n2)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.68
ALDH1A1 P00352 1/20 0.68
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
GABRA1 P14867 1/20 0.68
HPGD P15428 1/20 0.68
GABRG2 P18507 1/20 0.68
GABRB3 P28472 1/20 0.68
GABRA5 P31644 1/20 0.68
GABRA3 P34903 1/20 0.68
GABRA2 P47869 1/20 0.68
HSD17B10 Q99714 1/20 0.68
TDP1 Q9NUW8 1/20 0.68
SMN1; SMN2 Q16637 5/20 0.62
BRD4 O60885 2/20 0.61
LIN28A Q9H9Z2 1/20 0.61
MEN1 O00255 1/20 0.53
LMNA P02545 1/20 0.53
KMT2A Q03164 1/20 0.53
NPC1 O15118 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11623112 0.85 KDM4E (0.65) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
SCHEMBL10389396 0.85 KDM4E (0.65) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
SCHEMBL31265357 0.85 KDM4E (0.65) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
SCHEMBL11628686 0.85 KDM4E (0.69) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
SCHEMBL11489169 0.83 KDM4E (0.65) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
SCHEMBL10389924 0.82 SMN1; SMN2 (0.71) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
Ci-218872 SCHEMBL29469726 0.81 KDM4E (1.00) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
Ci-218872 SCHEMBL1320758 0.81 KDM4E (1.00) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
SCHEMBL15024914 0.80 KDM4E (0.83) KDM4EALDH1A1CYP1A2CYP3A4GABRA1
SCHEMBL10389919 0.79 SMN1; SMN2 (0.67) KDM4EALDH1A1CYP1A2CYP3A4GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4112095-A 6-Phenyl-1,2,4-triazolo[4,3-b]pyridazine hypotensive agents AMERICAN CYANAMID COMPANY (US) 1978-09-05 US disclosed