SCHEMBL11690331

SCHEMBL11690331

CCOC(=O)/C(=C\c1ccco1)C(C)=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.63
POLB P06746 4/20 0.63
ALDH1A1 P00352 5/20 0.52
MAPT P10636 13/20 0.50
MEN1 O00255 9/20 0.50
KMT2A Q03164 9/20 0.50
KDM4E B2RXH2 4/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
GLO1 Q04760 2/20 0.49
HPGD P15428 2/20 0.48
HSP90AA1 P07900 1/20 0.48
USP2 O75604 1/20 0.47
IDE P14735 1/20 0.47
TNNI3 P19429 1/20 0.47
TNNT2 P45379 1/20 0.47
TNNC1 P63316 1/20 0.47
NPSR1 Q6W5P4 4/20 0.45
LMNA P02545 4/20 0.45
PKM P14618 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10377521 1.00 TDP1 (0.63) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL20176814 1.00 TDP1 (0.63) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL11781592 0.92 POLB (0.68) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL11772644 0.88 TDP1 (0.63) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL27852160 0.88 TDP1 (0.63) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL11097979 0.85 POLB (0.66) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL11097975 0.85 POLB (0.66) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL22697045 0.85 POLB (0.66) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL9776425 0.85 POLB (0.59) TDP1POLBALDH1A1MAPTMEN1
SCHEMBL10988551 0.85 MAPT (0.47) TDP1POLBALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116287032-A Method for preparing 3-oxo-ethyl butyrate derivative by reacting aromatic aldehyde with ethyl acetoacetate under enzyme catalysis 岭南师范学院 2023-06-23 CN disclosed
US-4053614-A 1,2-PENTAMETHYLENE-1,4-DIHYDROPYRIDINE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DT) 1977-10-11 US disclosed
US-4024261-A HYPERTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-05-17 US disclosed
US-4022898-A ANTIHYPERTENSIVE AGENTS, VASODILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-05-10 US disclosed
US-4004015-A Bicyclic derivatives of 1,4-dihydropyridine as antihypertensive agents and coronary vessel dilators BAYER AKTIENGESELLSCHAFT (DT) 1977-01-18 US disclosed
US-4001258-A HYPOTENSIVES, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-01-04 US disclosed
US-4001235-A HYPOTENSIVES, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-01-04 US disclosed
US-3971791-A VASODILATION, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DT) 1976-07-27 US disclosed
US-3971790-A VASODILATION, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DT) 1976-07-27 US disclosed
US-3951994-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-20 US disclosed
US-3951988-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-20 US disclosed
US-3948923-A HYPOTENSIVE, VASODILATION BAYER AKTIENGESELLSCHAFT (DT) 1976-04-06 US disclosed
US-3946026-A HYPOTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-03-23 US disclosed
US-3939171-A HYPOTENSIVE, VASODILATION BAYER AKTIENGESELLSCHAFT (DT) 1976-02-17 US disclosed
US-3935220-A VASODILATION, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DT) 1976-01-27 US disclosed
US-3935223-A 2-Amino-1,4-dihydropyridine derivatives BAYER AKTIENGESELLSCHAFT (DT) 1976-01-27 US disclosed