Ridogrel

Ridogrel

SCHEMBL11708

O=C(O)CCCCO/N=C(\c1cccnc1)c1cccc(C(F)(F)F)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 19/20 1.00
TBXAS1 P24557 12/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ridogrel SCHEMBL30206884 1.00 TBXA2R (1.00) TBXA2RTBXAS1
Ridogrel SCHEMBL31639193 1.00 TBXA2R (1.00) TBXA2RTBXAS1
Ridogrel SCHEMBL11709 1.00 TBXA2R (1.00) TBXA2RTBXAS1
Ridogrel SCHEMBL11710 1.00 TBXA2R (1.00) TBXA2RTBXAS1
Ridogrel SCHEMBL7564456 0.99 TBXA2R (0.98) TBXA2RTBXAS1
Ridogrel SCHEMBL7564452 0.99 TBXA2R (0.98) TBXA2RTBXAS1
Ridogrel SCHEMBL27520191 0.99 TBXA2R (0.98) TBXA2RTBXAS1
SCHEMBL13933082 0.87 TBXA2R (0.77) TBXA2RTBXAS1
SCHEMBL9601449 0.87 TBXA2R (0.76) TBXA2RTBXAS1
SCHEMBL9601444 0.87 TBXA2R (0.76) TBXA2RTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2426 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025184468-A9 MEASUREMENT OF URINE THROMBOXANE METABOLITES TO PREDICT SURVIVAL UNIVERSITY OF MASSACHUSETTS (US) 2025-10-16 WO claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20250120908-A1 ORAL FILM FORMULATION FOR MODULATING ABSORPTION PROFILE INTELGENX CORP. (CA) 2025-04-17 US claimed
US-12156937-B2 Oral film formulation for modulating absorption profile INTELGENX CORP. (CA) 2024-12-03 US claimed
US-20230047314-A1 ORAL FILM FORMULATION FOR MODULATING ABSORPTION PROFILE INTELGENX CORP. (CA) 2023-02-16 US claimed
US-11471406-B2 Oral film formulation for modulating absorption profile INTELGENX CORP. (CA) 2022-10-18 US claimed
US-20210022991-A1 ORAL FILM FORMULATION FOR MODULATING ABSORPTION PROFILE INTELGENX CORP. (CA) 2021-01-28 US claimed
US-10828254-B2 Oral film formulation for modulating absorption profile INTELGENX CORP. (CA) 2020-11-10 US claimed
CN-107049932-B Small molecule drug in-situ phase change gel sustained release system and preparation method thereof 四川大学 2020-11-06 CN claimed
EP-3643298-A1 IN SITU PHASE CHANGE GEL SUSTAINED-RELEASE SYSTEM FOR SMALL MOLECULE DRUG AND PREPARATION METHOD THEREOF Sichuan University (CN) 2020-04-29 EP claimed
CN-1179716-A Low dose ridogrel formulations and their use for treatment of inflammatory bowel diseases JANSSEN PHARMACEUTICA NV (BE) 1998-04-22 CN claimed
WO-1998015265-A1 COLONIC DELIVERY OF WEAK ACID DRUGS DANBIOSYST UK LIMITED (GB) 1998-04-16 WO claimed
EP-0817631-A2 LOW DOSE RIDOGREL FORMULATIONS AND THEIR USE FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASES JANSSEN PHARMACEUTICA N.V. (BE) 1998-01-14 EP claimed
WO-1996030016-A2 LOW DOSE RIDOGREL FORMULATIONS AND THEIR USE FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASES JANSSEN PHARMACEUTICA N.V. (BE) 1996-10-03 WO claimed
WO-1996017606-A1 USE OF INFLAMMATORY MODULATORS IN THE TREATMENT OF CHRONIC OR RECALCITRANT SKIN DAMAGE BRISTOL-MYERS SQUIBB COMPANY (US) 1996-06-13 WO claimed
EP-0221601-B1 [[[(3-Pyridinyl)methylen]amino]oxy]alkanoic acids and esters JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-10 EP claimed
WO-1992019182-A2 METHOD OF ATTENUATION OF NEOINTIMAL PROLIFERATION BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1992-11-12 WO claimed
US-4963573-A INHIBIT BIOSYNTHESIS OF THROMBOXANE A2 JANSSEN PHARMACEUTICA N.V. (BE) 1990-10-16 US claimed
US-4746671-A THROMBOXANE SYNTHETASE INHIBITION JANSSEN PHARMACEUTICA N.V. (BE) 1988-05-24 US claimed
EP-0221601-A1 [[[(3-Pyridinyl)methylen]amino]oxy]alkanoic acids and esters JANSSEN PHARMACEUTICA N.V. (BE) 1987-05-13 EP claimed