SCHEMBL11740657

SCHEMBL11740657

O=C(O)Cc1ccc2c(Cl)cccc2c1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.60
THRA P10827 1/20 0.55
THRB P10828 1/20 0.55
CA2 P00918 1/20 0.53
SLC22A12 Q96S37 11/20 0.50
GAA P10253 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
PTGS1 P23219 1/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11462511 0.87 AKR1B1 (0.56) AKR1B1THRATHRBCA2SLC22A12
SCHEMBL21585558 0.81 AKR1B1 (0.62) AKR1B1THRATHRBCA2GAA
SCHEMBL30496795 0.81 TDP1 (0.66) AKR1B1THRATHRBSLC22A12GAA
SCHEMBL10343028 0.81 AKR1B1 (0.58) AKR1B1THRATHRBCA2GAA
SCHEMBL31074301 0.80 AKR1B1 (0.60) AKR1B1THRATHRBSLC22A12GAA
SCHEMBL11740239 0.80 AKR1B1 (0.60) AKR1B1THRATHRBSLC22A12GAA
SCHEMBL27537426 0.80 AKR1B1 (0.60) AKR1B1THRATHRBGAANR1H4
SCHEMBL30557996 0.79 AKR1B1 (0.84) AKR1B1SLC22A12GAANR1H4PTGS1
SCHEMBL15352237 0.79 CYP1A2 (0.48) AKR1B1THRATHRBMEN1ALDH1A1
SCHEMBL10392245 0.79 CYP1A2 (0.48) AKR1B1THRATHRBCA2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4045485-A ANTIINFLAMMATORY, ANALGESIC, ANTIPYRETIC AND ANTIPRURITIC ACTIVITY SYNTEX CORPORATION (US) 1977-08-30 US disclosed
US-3960936-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIPYRETICS, SKIN DISORDERS SYNTEX CORPORATION (PM) 1976-06-01 US disclosed
US-3947472-A ANTIINFLAMMATORY, ANALGESIC, ANTIPYRETIC, ANTIPRURITIC SYNTEX CORPORATION (PM) 1976-03-30 US disclosed
US-3935273-A ANTIINFLAMMATORY, ANALGESIC, ANTIPYRETIC, ANTIPRURITIC SYNTEX CORPORATION (US) 1976-01-27 US disclosed