SCHEMBL11814264

SCHEMBL11814264

Clc1cc2ccccc2c(-n2ccnc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 12/20 0.52
CYP1A2 P05177 11/20 0.52
LMNA P02545 10/20 0.52
CYP2D6 P10635 10/20 0.52
CYP2C19 P33261 10/20 0.52
CLK4 Q9HAZ1 7/20 0.52
MEN1 O00255 6/20 0.52
KMT2A Q03164 6/20 0.52
USP2 O75604 5/20 0.52
HSD17B10 Q99714 4/20 0.52
TP53 P04637 4/20 0.52
CYP11B1 P15538 3/20 0.47
CYP11B2 P19099 3/20 0.47
CYP19A1 P11511 2/20 0.47
TDP1 Q9NUW8 4/20 0.46
MAPT P10636 2/20 0.46
HIF1A Q16665 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 1/20 0.45
IDO1 P14902 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11814515 0.81 CYP3A4 (0.52) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL11820505 0.79 CYP3A4 (0.53) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL11820482 0.78 CYP3A4 (0.46) CYP3A4CYP1A2LMNACYP2D6CYP2C19
Hydrochloric Acid SCHEMBL11819489 0.77 CYP3A4 (0.45) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL11814063 0.76 CYP3A4 (0.44) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL7646271 0.76 COMT (0.52) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL14300759 0.75 CYP3A4 (0.67) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL15688941 0.75 CYP11B1 (0.54) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL14103054 0.75 DHODH (0.48) CYP3A4CYP1A2LMNACYP2D6CYP2C19
SCHEMBL11816276 0.74 CYP3A4 (0.51) CYP3A4CYP1A2LMNACYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3961062-A Pharmaceutical composition containing 1-(imidazole-1-yl)-isoquinolines and method of treating hyperlipemia HOECHST AKTIENGESELLSCHAFT (DT) 1976-06-01 US claimed
US-3961062-A Pharmaceutical composition containing 1-(imidazole-1-yl)-isoquinolines and method of treating hyperlipemia HOECHST AKTIENGESELLSCHAFT (DT) 1976-06-01 US disclosed