SCHEMBL11845293

SCHEMBL11845293

O=C1c2ccccc2N(Cc2ccc(Cl)cc2)C2=NCCN12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 1.00
HTT P42858 4/20 0.60
GAA P10253 1/20 0.58
GFER P55789 1/20 0.58
CES2 O00748 1/20 0.56
BCHE P06276 1/20 0.56
CES1 P23141 1/20 0.56
KMT2A Q03164 3/20 0.55
TP53 P04637 2/20 0.55
PRKAG1 P54619 3/20 0.52
PRKAB1 Q9Y478 3/20 0.52
PRKAA1 Q13131 2/20 0.52
DRD2 P14416 1/20 0.49
DRD4 P21917 1/20 0.49
SOS1 Q07889 1/20 0.48
MEN1 O00255 2/20 0.48
LMNA P02545 3/20 0.47
PRKAA2 P54646 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11850062 0.93 TSHR (0.86) TSHRHTTGAAGFERCES2
SCHEMBL2493279 0.91 TSHR (0.83) TSHRHTTGAAGFERCES1
SCHEMBL11847278 0.89 TSHR (0.80) TSHRHTTGAAGFERKMT2A
SCHEMBL11842852 0.89 TSHR (0.80) TSHRHTTGAAGFERKMT2A
Hydrochloric Acid SCHEMBL11845788 0.88 TSHR (0.78) TSHRHTTGAAGFERKMT2A
SCHEMBL11855278 0.86 TSHR (0.75) TSHRHTTGAAGFERCES2
SCHEMBL11850001 0.85 TSHR (0.74) TSHRHTTGAAGFERKMT2A
Hydrochloric Acid SCHEMBL11851095 0.85 TSHR (0.73) TSHRHTTGAAGFERKMT2A
SCHEMBL11849241 0.84 TSHR (0.72) TSHRHTTGAAGFERKMT2A
SCHEMBL11838764 0.84 TSHR (0.72) TSHRHTTGAAGFERKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3969506-A BRONCHODILATOR SANDOZ, INC. (US) 1976-07-13 US claimed
US-3969506-A BRONCHODILATOR SANDOZ, INC. (US) 1976-07-13 US disclosed