SCHEMBL11859249

SCHEMBL11859249

O=CNCC1c2ccccc2C=Cc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.50
HRH1 P35367 3/20 0.45
CYP2D6 P10635 3/20 0.45
KDM4E B2RXH2 2/20 0.45
LMNA P02545 2/20 0.45
CYP3A4 P08684 2/20 0.45
TP53 P04637 1/20 0.45
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
DRD2 P14416 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
NFKB1 P19838 1/20 0.45
CHRM3 P20309 1/20 0.45
SLC6A2 P23975 1/20 0.45
HTR2C P28335 1/20 0.45
ADRA1A P35348 1/20 0.45
DRD3 P35462 1/20 0.45
THPO P40225 1/20 0.45
OPRK1 P41145 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11865510 0.87 HTR2A (0.39) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL11859798 0.87 KDM4E (0.39) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL11857247 0.83 HTR2A (0.38) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL11863543 0.83 P2RX4 (0.37) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL11868591 0.83 HTR2A (0.37) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL11869992 0.82 HTR2A (0.36) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL1509217 0.81 HTR2A (0.47) HTR2AHRH1KMT2AADH1BADH1C
SCHEMBL11868581 0.80 TACR1 (0.36) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL11861536 0.79 TSHR (0.38) HTR2AHRH1CYP2D6KDM4ELMNA
SCHEMBL11857446 0.75 HTR2A (0.62) HTR2AHRH1CYP2D6KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3992445-A ANTICONVULSANTS MERCK & CO., INC. (US) 1976-11-16 US claimed
US-3992445-A ANTICONVULSANTS MERCK & CO., INC. (US) 1976-11-16 US disclosed
US-3992445-A ANTICONVULSANTS MERCK & CO., INC. (US) 1976-11-16 US disclosed