SCHEMBL11890901

SCHEMBL11890901

CN1CCOc2c(Cl)nn3c(Br)nnc3c21

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 15/20 0.32
PIM3 Q86V86 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2176774 0.89 PIM1 (0.36) PIM1PIM3
SCHEMBL27083001 0.78
SCHEMBL12492784 0.75 PIM1 (0.57) PIM1PIM3
SCHEMBL2175236 0.75
SCHEMBL2176239 0.74 PIM1 (0.58) PIM1PIM3
SCHEMBL11299291 0.72 HTT (0.40) PIM1
SCHEMBL14554064 0.70 PIM1 (0.31) PIM1
SCHEMBL14554041 0.69
SCHEMBL14485343 0.68
SCHEMBL27081681 0.67 CSNK1E (0.37) PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012098387-A1 6, 7-RING-FUSED TRIAZOLO [4, 3 - B] PYRIDAZINE DERIVATIVES AS PIM INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-07-26 WO disclosed