Dihydrocapsaicin

Dihydrocapsaicin

SCHEMBL119080

COc1cc(CNC(=O)CCCCCCC(C)C)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 1.00
CYP3A4 P08684 5/20 1.00
CYP2D6 P10635 4/20 1.00
CYP2C9 P11712 3/20 1.00
CYP2C19 P33261 3/20 1.00
MEN1 O00255 3/20 1.00
KMT2A Q03164 3/20 1.00
BLM P54132 2/20 1.00
PMP22 Q01453 2/20 1.00
POLB P06746 1/20 1.00
TSHR P16473 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
HDAC3 O15379 1/20 0.80
HDAC4 P56524 1/20 0.80
HDAC1 Q13547 1/20 0.80
HDAC7 Q8WUI4 1/20 0.80
HDAC2 Q92769 1/20 0.80
HDAC10 Q969S8 1/20 0.80
HDAC11 Q96DB2 1/20 0.80
HDAC8 Q9BY41 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9059706 1.00 CYP1A2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1870592 1.00 CYP1A2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
Dihydrocapsaicin SCHEMBL29819467 1.00 CYP1A2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL117622 1.00 CYP1A2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL29425544 1.00 CYP1A2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5348698 0.91 CYP1A2 (0.90) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
Dihydrocapsaicin SCHEMBL28311536 0.91 CYP1A2 (0.82) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL17778309 0.90 CYP1A2 (0.82) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL17778308 0.90 CYP1A2 (0.82) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL1703135 0.90 CYP1A2 (0.81) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5174 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4210687-B1 TRPV1 AGONISTS IN THE PREVENTION OF DIABETIC ULCERS IMPERIAL COLLEGE INNOVATIONS LTD (GB) 2026-05-27 EP claimed
CN-122060791-A Application of ERF/AP2 transcription factor CcADAP in regulation and control of peppery degree of peppery peppers 浙江大学海南研究院 2026-05-19 CN claimed
EP-4683527-A1 VAPORIZABLE ALKALOID COMPOSITIONS AND METHODS OF USE THEREOF Ready Mix Naturals, LLC (US) 2026-01-28 EP claimed
EP-4680210-A1 MEDICAL PATCH COMPRISING SKIN IRRITATING ACTIVE AGENT LTS Lohmann Therapie-Systeme AG (DE) 2026-01-21 EP claimed
US-12497381-B2 Vaporizable alkaloid compositions and methods of use thereof Ready Mix Naturals, LLC (US) 2025-12-16 US claimed
US-12478091-B2 Vaporizable alkaloid compositions and methods of use thereof Ready Mix Naturals, LLC (US) 2025-11-25 US claimed
US-20250325533-A1 TRYPTAMINE COMPOSITIONS FOR ENHANCING NEURITE OUTGROWTH TURTLE BEAR HOLDINGS LLC (US) 2025-10-23 US claimed
US-12440839-B2 High-throughput system and method for the temporary permeabilization of cells using lipid bilayers THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-10-14 US claimed
EP-4606437-A1 COSMETIC COMPOSITIONS TO INHIBIT THE ACTIVITY OF KLF4, TO REDUCE SKIN, HAIR, MUCOUS MEMBRANES AGING LABORATOIRE NATIVE (FR) 2025-08-27 EP claimed
EP-4599698-A1 PRODUCTS COMPRISING SENSORY AGENTS Nicoventures Trading Limited (GB) 2025-08-13 EP claimed
US-5672354-A Treated bird seed preferentially palatable to birds but not palatable to animals having capsaicin sensitive receptors THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 1997-09-30 US claimed
WO-1997002273-A1 WARMING COMPOUNDS THE PROCTER & GAMBLE COMPANY (US) 1997-01-23 WO claimed
WO-1996040079-A1 METHOD AND COMPOSITIONS FOR CONTROLLING ORAL AND PHARYNGEAL PAIN USING CAPSAICINOIDS EMORY UNIVERSITY (US) 1996-12-19 WO claimed
EP-0723948-A1 Capsaicinoid lachrymator Defense Technology Corporation of America (US) 1996-07-31 EP claimed
US-5397385-A Anti-fouling coating composition containing capsaicin GEORGES, PETER J. 1995-03-14 US claimed
WO-1994008840-A1 MARINE ORGANISM REPELLENT FOR PROTECTING UNDERWATER OBJECTS FISCHER KENNETH J (US) 1994-04-28 WO claimed
WO-1993023061-A1 THERAPEUTIC USES OF PUNGENT BOTANICALS AND THEIR RELATED COMPOUNDS STAGGS JEFF J (US) 1993-11-25 WO claimed
EP-0546078-A4 BIRDFOOD CONTAINING CAPSAICIN OR ITS DERIVATIVES OR ANALOGUES US HEALTH (US) 1993-09-15 EP claimed
EP-0546078-A1 BIRDFOOD CONTAINING CAPSAICIN OR ITS DERIVATIVES OR ANALOGUES THE UNITED STATES OF AMERICA as represented by the Secretary UNITED STATES DEPARTMENT OF COMMERCE (US) 1993-06-16 EP claimed
WO-1992003923-A1 BIRDFOOD CONTAINING CAPSAICIN OR ITS DERIVATIVES OR ANALOGUES THE UNITED STATES OF AMERICA, represented by THE SCRETARY, UNITED STATES DEPARTMENT OF COMMERCE (US) 1992-03-19 WO claimed