SCHEMBL12031803

SCHEMBL12031803

Cc1ccccc1C(=O)N[C@H](C(=O)N1CCC[C@H]1C=O)C(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 6/20 0.55
ACE P12821 2/20 0.45
STAT6 P42226 4/20 0.45
ELANE P08246 2/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CCR8 P51685 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM2 P08172 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8289016 0.90 CCR1 (0.49) CCR1ACESTAT6ELANE
SCHEMBL12031884 0.88 CCR1 (0.47) CCR1STAT6ELANE
SCHEMBL12949865 0.86 CCR1 (0.41) CCR1STAT6ELANECHRM2
SCHEMBL8286865 0.85 CCR1 (0.46) CCR1STAT6ELANERAB9A
SCHEMBL14181582 0.85 STAT6 (0.42) CCR1STAT6ELANE
SCHEMBL3183987 0.84 ACE (0.57) CCR1ACESTAT6ELANE
SCHEMBL12031887 0.84 CCR1 (0.43) CCR1STAT6ELANE
SCHEMBL8288841 0.84 CCR1 (0.43) CCR1STAT6ELANE
SCHEMBL12031332 0.83 CCR1 (0.49) CCR1ACESTAT6ELANENPC1
SCHEMBL12031752 0.83 STAT6 (0.43) CCR1STAT6ELANENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399915-A1 Process and intermediates for the preparation of aspartic acetal caspase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-12-28 EP disclosed