SCHEMBL12068435

SCHEMBL12068435

N[C@@H](C(=O)N1CCC[C@H]1c1ncc(-c2ccc(C#Cc3ccc(-c4cnc([C@@H]5CCCN5C(=O)[C@H](NC(=O)N5CCC[C@@H]5CO)c5ccccc5)[nH]4)cc3)cc2)[nH]1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.48
CYP3A4 P08684 4/20 0.45
CYP2C9 P11712 3/20 0.45
NR1I2 O75469 1/20 0.45
ABCB11 O95342 1/20 0.45
OPRK1 P41145 1/20 0.45
OPRM1 P35372 2/20 0.45
OPRD1 P41143 2/20 0.45
CYP1A2 P05177 2/20 0.45
PRCP P42785 8/20 0.43
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12068434 1.00 KCNH2 (0.48) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL12068443 0.92 KCNH2 (0.51) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL10145305 0.91 KCNH2 (0.57) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL10145302 0.91 KCNH2 (0.57) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL13293088 0.90 KCNH2 (0.48) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL12066429 0.89 KCNH2 (0.48) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL10176518 0.88 KCNH2 (0.47) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL13293010 0.88 KCNH2 (0.47) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL10176641 0.88 KCNH2 (0.49) KCNH2CYP3A4CYP2C9NR1I2ABCB11
SCHEMBL13293353 0.87 KCNH2 (0.46) KCNH2CYP3A4CYP2C9NR1I2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011150243-A1 INHIBITORS OF HCV NS5A PRESIDIO PHARMACEUTICALS, INC. (US) 2011-12-01 WO disclosed
WO-2010065668-A1 INHIBITORS OF HCV NS5A PRESIDIO PHARMACEUTICALS, INC. (US) 2010-06-10 WO disclosed