SCHEMBL12150720

SCHEMBL12150720

Cc1nc(Cl)c(/C=C/c2ccccc2F)c(N[C@@H]2C[C@H](CO)[C@@H](O)C2)n1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NAE1 Q13564 5/20 0.35
UBA3 Q8TBC4 5/20 0.35
NFE2L2 Q16236 4/20 0.33
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12150570 0.89 IRAK4 (0.38) NAE1UBA3NFE2L2KMT2A
SCHEMBL12150685 0.85 IRAK4 (0.42)
SCHEMBL12150694 0.79 IRAK4 (0.40)
SCHEMBL802894 0.76 PDE10A (0.39) NAE1UBA3
SCHEMBL802501 0.76 PDE10A (0.39) NAE1UBA3
SCHEMBL12150716 0.75 IRAK4 (0.43)
SCHEMBL12150673 0.75 IRAK4 (0.43)
SCHEMBL12150542 0.75 IRAK4 (0.54)
SCHEMBL12150681 0.70 IRAK4 (0.39)
SCHEMBL12150672 0.70 IRAK4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110286965-A1 ETHENYL-SUBSTITUTED PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATING VIRAL INFECTIONS MERCK SHARP & DOHME LLC 2011-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110286965-A1 ETHENYL-SUBSTITUTED PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATING VIRAL INFECTIONS CYP2C9, PNP, UGT1A3 NAE1 719/4885UBA3 203/4885NFE2L2 2307/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.