SCHEMBL12152007

SCHEMBL12152007

O=Cc1c[nH]c2c(-n3ccnn3)ncc(F)c12

nearest known ligand 0.35

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10326904 0.82 CYP3A4 (0.34) NOTUM
SCHEMBL1733111 0.77 NOTUM (0.33) NOTUM
SCHEMBL13411361 0.77 CYP1A2 (0.38)
SCHEMBL12151881 0.76 NOTUM (0.33) NOTUM
SCHEMBL12528172 0.74 CYP3A4 (0.34) NOTUM
SCHEMBL13909729 0.71 KMT2A (0.32)
SCHEMBL13909691 0.71 CYP2A6 (0.38)
SCHEMBL9286142 0.71 CYP3A4 (0.39)
Hydrochloric Acid SCHEMBL9284226 0.70 CYP3A4 (0.39)
SCHEMBL2628936 0.69 NOTUM (0.41) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012142080-A1 THIOAMIDE, AMIDOXIME AND AMIDRAZONE DERIVATIVES AS HIV ATTACHMENT INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-10-18 WO disclosed
EP-1943221-B1 PIPERAZINE AMIDINES AS ANTIVIRAL AGENTS BRISTOL MYERS SQUIBB CO (US) 2011-11-23 EP disclosed
US-7807671-B2 Diketo-piperazine and piperidine derivatives as antiviral agents BRISTOL-MYERS SQUIBB COMPANY (US) 2010-10-05 US disclosed