SCHEMBL12166181

SCHEMBL12166181

COCCN(C)C(=O)N1CCN(Cc2cc3nc(-c4cccc(O)c4)nc(N)c3s2)CC1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 15/20 0.52
PIK3CD O00329 9/20 0.48
PIK3CB P42338 8/20 0.48
PIK3CG P48736 8/20 0.48
ADORA2A P29274 4/20 0.42
ADORA1 P30542 3/20 0.39
PARP1 P09874 1/20 0.37
MTOR P42345 1/20 0.37
PARP2 Q9UGN5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL190794 0.87 PIK3CA (0.71) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL17255576 0.77 PIK3CA (0.69) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL958777 0.76 PIK3CA (0.78) PIK3CAPIK3CDPIK3CBPIK3CGPARP1
SCHEMBL1180282 0.76 PIK3CA (0.69) PIK3CAPIK3CDPIK3CBPIK3CGPARP1
SCHEMBL1180888 0.76 PIK3CA (0.66) PIK3CAPIK3CDPIK3CBPIK3CGPARP1
SCHEMBL1180666 0.73 PIK3CA (0.56) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL964128 0.72 PIK3CA (0.75) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL12166175 0.72 PIK3CA (0.57) PIK3CAPIK3CDPIK3CBPIK3CGADORA2A
SCHEMBL962251 0.72 PIK3CA (0.73) PIK3CAPIK3CDPIK3CBPIK3CG
SCHEMBL960842 0.72 PIK3CA (0.82) PIK3CAPIK3CDPIK3CBPIK3CGMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041139-B1 PHARMACEUTICAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2011-11-09 EP disclosed