SCHEMBL12166394

SCHEMBL12166394

CS(=O)(=O)Nc1cccc(-c2nc(NCCO)c3sc(CN4CCN(S(C)(=O)=O)CC4)cc3n2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.55
PIK3CD O00329 9/20 0.55
PIK3CB P42338 8/20 0.55
PIK3CG P48736 8/20 0.55
CYP1A2 P05177 5/20 0.51
CYP3A4 P08684 5/20 0.51
MAPK1 P28482 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
MTOR P42345 6/20 0.46
USP2 O75604 4/20 0.46
CYP2C19 P33261 4/20 0.46
CLK4 Q9HAZ1 4/20 0.46
CYP2D6 P10635 3/20 0.46
ALOX15 P16050 2/20 0.46
ALDH1A1 P00352 2/20 0.46
APEX1 P27695 1/20 0.46
CASP7 P55210 1/20 0.46
ABCC4 O15439 1/20 0.44
ABCB11 O95342 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12166180 0.89 PIK3CA (0.69) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL12166291 0.87 PIK3CA (0.54) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL10265724 0.82 PIK3CA (0.79) PIK3CAPIK3CDPIK3CBPIK3CGCYP1A2
SCHEMBL12166377 0.79 ABCC4 (0.48) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL12166214 0.76 PIK3CA (0.56) PIK3CAPIK3CDPIK3CBPIK3CGCYP1A2
SCHEMBL190300 0.72 PIK3CA (0.80) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL12166370 0.72 PIK3CA (0.59) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL190409 0.71 PIK3CA (1.00) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL8212241 0.71 PIK3CA (0.74) PIK3CAPIK3CDPIK3CBPIK3CGMTOR
SCHEMBL962660 0.70 PIK3CA (1.00) PIK3CAPIK3CDPIK3CBPIK3CGMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041139-B1 PHARMACEUTICAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2011-11-09 EP disclosed