SCHEMBL12192092

SCHEMBL12192092

CC(=O)/C(C)=C/c1ccc2nc(C(C)(C)NC(=O)c3ccc4c(C5CCCC5)c(-c5ccc(F)cn5)n(C)c4c3)n(C)c2c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.56
CTSG P08311 1/20 0.56
MAOA P21397 1/20 0.56
DRD1 P21728 1/20 0.56
CYP3A4 P08684 12/20 0.53
CYP2C19 P33261 11/20 0.53
KCNH2 Q12809 1/20 0.49
CYP2C9 P11712 3/20 0.46
CYP2D6 P10635 2/20 0.46
CYP1A2 P05177 2/20 0.41
CYP2C8 P10632 1/20 0.39
SCN9A Q15858 3/20 0.39
ACSS2 Q9NR19 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12922282 0.95 HTR2A (0.57) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12192094 0.92 CYP3A4 (0.60) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12922293 0.87 CYP3A4 (0.61) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12192090 0.85 CYP3A4 (0.53) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12899620 0.85 CYP3A4 (0.58) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12192129 0.85 KCNH2 (0.48) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12192098 0.81 CYP3A4 (0.54) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12922286 0.81 CYP3A4 (0.54) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL15109267 0.80 CYP3A4 (0.59) HTR2ACTSGMAOADRD1CYP3A4
SCHEMBL12922309 0.80 KCNH2 (0.49) HTR2ACTSGMAOADRD1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030309-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-04 US disclosed