SCHEMBL12192142

SCHEMBL12192142

COc1ccc(-c2c(C3CCCC3)c3ccc(C(=O)NC4(c5nc6ccc(/C=C/C(C)=O)cc6n5C)CCC4)cc3n2C)nn1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.57
CYP2C8 P10632 1/20 0.57
CYP3A4 P08684 15/20 0.51
CYP2C19 P33261 14/20 0.51
CYP2C9 P11712 3/20 0.47
KCNH2 Q12809 1/20 0.45
CYP2D6 P10635 1/20 0.41
CTSG P08311 1/20 0.40
MAOA P21397 1/20 0.40
DRD1 P21728 1/20 0.40
HTR2A P28223 1/20 0.40
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12922321 0.95 CYP1A2 (0.59) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL12899644 0.92 CYP1A2 (0.57) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL13680382 0.88 CYP1A2 (0.68) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL12899592 0.87 CYP1A2 (0.58) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL12899654 0.87 CYP3A4 (0.53) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL13680359 0.87 CYP3A4 (0.64) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL13680358 0.87 CYP3A4 (0.63) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL13680361 0.87 CYP1A2 (0.61) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL13680370 0.86 CYP3A4 (0.63) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9
SCHEMBL13680369 0.86 CYP3A4 (0.63) CYP1A2CYP2C8CYP3A4CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030309-B2 Viral polymerase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-04 US disclosed