SCHEMBL12202085

SCHEMBL12202085

C/C(=C\C(C(C)C)N(C)C(=O)C(NC(=O)C1CCCCCN1C)C(C)(C)C)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.60
ELANE P08246 3/20 0.35
STAT6 P42226 4/20 0.33
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
HDAC1 Q13547 1/20 0.31
CASP1 P29466 1/20 0.30
CASP4 P49662 1/20 0.30
CASP5 P51878 1/20 0.30
CASP7 P55210 1/20 0.30
CASP9 P55211 1/20 0.30
CASP8 Q14790 1/20 0.30
CASP10 Q92851 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14592521 1.00 TUBB1 (0.60) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL58979 1.00 TUBB1 (0.60) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL16316203 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL18421085 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL18421084 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL58832 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL13681898 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL13681981 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL89591 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6
SCHEMBL14592398 0.99 TUBB1 (0.59) TUBB1ELANESTAT6CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2374454-A1 Hemiasterlin derivatives and uses thereof in the treatment of cancer Eisai R&D Management Co., Ltd. (JP) 2011-10-12 EP disclosed