SCHEMBL12246720

SCHEMBL12246720

[C-]#[N+]c1cccc(-c2ccc3c(c2)/C(=N/C#N)CC2(CCCc4ccccc4C2)O3)c1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.35
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12246644 0.95 BACE1 (0.38) BACE1SLC6A2SLC6A4SLC6A3
SCHEMBL12246655 0.92 BACE1 (0.33) BACE1SLC6A2SLC6A4SLC6A3
SCHEMBL1820029 0.86 BACE1 (0.45) BACE1
SCHEMBL1820031 0.86 BACE1 (0.45) BACE1
SCHEMBL12246718 0.83 KDM4E (0.41) BACE1SLC6A2SLC6A4SLC6A3
SCHEMBL2374775 0.81 BACE1 (0.44) BACE1
SCHEMBL2374777 0.81 BACE1 (0.44) BACE1
SCHEMBL12247524 0.81 USP2 (0.31) BACE1SLC6A2SLC6A4SLC6A3
SCHEMBL7962670 0.80 BACE1 (0.35) BACE1
SCHEMBL12246645 0.78 BACE1 (0.41) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8921359-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2014-12-30 US disclosed
US-8450308-B2 Inhibitors of beta-secretase VITAE PHARMACEUTICALS, INC. (US) 2013-05-28 US disclosed
US-20110218192-A1 Inhibitors Of Beta-Secretase VITAE PHARMACEUTICALS, INC. (US) 2011-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110218192-A1 Inhibitors Of Beta-Secretase BACE1, BACE2, APP BACE1 1/4885SLC6A2 819/4885SLC6A4 2071/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.