SCHEMBL12281952

SCHEMBL12281952

CN(C)CCCS(=O)(=O)c1cccc(-c2n[nH]c3ccc(NC(=O)C(c4ccsc4)N4CCCC4)cc23)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTK P33981 17/20 0.74
AURKB Q96GD4 6/20 0.74
AURKA O14965 5/20 0.74
PLK4 O00444 3/20 0.74
CHEK2 O96017 3/20 0.74
CYP3A4 P08684 3/20 0.74
CYP2C9 P11712 3/20 0.74
CYP1A1 P04798 2/20 0.74
CYP1A2 P05177 2/20 0.74
CYP2E1 P05181 2/20 0.74
CYP2C8 P10632 2/20 0.74
CYP2D6 P10635 2/20 0.74
CYP2A6 P11509 2/20 0.74
CYP4B1 P13584 2/20 0.74
CYP2B6 P20813 2/20 0.74
CYP3A5 P20815 2/20 0.74
CYP2A7 P20853 2/20 0.74
CYP3A7 P24462 2/20 0.74
CYP2F1 P24903 2/20 0.74
CYP2C18 P33260 2/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15476743 0.83 TTK (0.61) TTKAURKBAURKAPLK4CHEK2
Trifluoroacetic Acid SCHEMBL2566375 0.81 TTK (0.90) TTKAURKBAURKAPLK4CHEK2
Trifluoroacetic Acid SCHEMBL2592428 0.81 TTK (0.90) TTKAURKBAURKAPLK4CHEK2
SCHEMBL15476598 0.81 TTK (0.62) TTKAURKBAURKAPLK4CHEK2
SCHEMBL12282488 0.81 TTK (0.65) TTKAURKBAURKAPLK4CHEK2
Trifluoroacetic Acid SCHEMBL2570005 0.81 TTK (0.89) TTKAURKBAURKAPLK4CHEK2
SCHEMBL14873402 0.79 TTK (0.71) TTKAURKBAURKAPLK4CHEK2
SCHEMBL14873430 0.78 TTK (0.69) TTKAURKBAURKAPLK4CHEK2
SCHEMBL14863660 0.78 TTK (0.69) TTKAURKBAURKAPLK4CHEK2
SCHEMBL20211279 0.76 TTK (0.69) TTKAURKBAURKAPLK4CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011123937-A1 KINASE INHIBITORS AND METHOD OF TREATING CANCER WITH SAME UNIVERSITY HEALTH NETWORK (CA) 2011-10-13 WO disclosed