SCHEMBL12285337

SCHEMBL12285337

Cn1cc(C2CCN(C(=O)OC(C)(C)C)CC2)c2ccc(Nc3ccc(F)c(F)c3)nc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.47
JAK2 O60674 9/20 0.44
JAK3 P52333 8/20 0.44
PTK2 Q05397 8/20 0.44
APP P05067 2/20 0.44
MAPT P10636 1/20 0.42
CNR1 P21554 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
GPR35 Q9HC97 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
JAK1 P23458 1/20 0.42
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41
THRB P10828 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TRPV3 Q8NET8 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12127997 0.92 GALR2 (0.49) SCN9AJAK2JAK3PTK2MAPT
SCHEMBL12284976 0.86 MAPT (0.49) SCN9AMAPTLMNATHRBTP53
SCHEMBL12128251 0.85 APP (0.62) SCN9AJAK2JAK3PTK2APP
SCHEMBL12129676 0.84 APP (0.55) JAK2APP
SCHEMBL12288140 0.83 SCN9A (0.46) SCN9AJAK2JAK3PTK2LMNA
SCHEMBL12131793 0.83 SCN9A (0.53) SCN9AAPP
SCHEMBL12128397 0.81 APP (0.53) SCN9AAPPMAPTTP53
SCHEMBL12128012 0.81 GALR2 (0.47) SCN9AJAK2JAK3PTK2MAPT
SCHEMBL12129153 0.79 APP (0.69) JAK2JAK3PTK2APP
SCHEMBL12127688 0.79 SCN9A (0.52) SCN9AJAK2JAK3MAPTJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011128455-A1 NOVEL COMPOUNDS FOR THE TREATMENT OF DISEASES ASSOCIATED WITH AMYLOID OR AMYLOID-LIKE PROTEINS AC IMMUNE S.A. (CH) 2011-10-20 WO disclosed