SCHEMBL12299260

SCHEMBL12299260

Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3N)s2)cc(N2CCN(CCO)CC2)n1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 14/20 0.83
SRC P12931 6/20 0.83
PKMYT1 Q99640 3/20 0.83
BCR P11274 3/20 0.83
EPHB6 O15197 2/20 0.83
EGFR P00533 2/20 0.83
LCK P06239 2/20 0.83
FYN P06241 2/20 0.83
CSF1R P07333 2/20 0.83
YES1 P07947 2/20 0.83
LYN P07948 2/20 0.83
RET P07949 2/20 0.83
HCK P08631 2/20 0.83
KIT P10721 2/20 0.83
BRAF P15056 2/20 0.83
EPHA1 P21709 2/20 0.83
EPHA2 P29317 2/20 0.83
EPHA3 P29320 2/20 0.83
EPHA8 P29322 2/20 0.83
EPHB2 P29323 2/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13378598 0.94 ABL1 (0.89) ABL1SRCPKMYT1BCREPHB6
SCHEMBL31634945 0.94 ABL1 (0.89) ABL1SRCPKMYT1BCREPHB6
SCHEMBL21350067 0.92 ABL1 (0.86) ABL1SRCPKMYT1BCREPHB6
SCHEMBL28426331 0.92 ABL1 (0.84) ABL1SRCPKMYT1BCREPHB6
SCHEMBL28427234 0.92 ABL1 (0.84) ABL1SRCPKMYT1BCREPHB6
SCHEMBL14153376 0.91 ABL1 (0.83) ABL1SRCPKMYT1BCREPHB6
Dasatinib Anhydrous SCHEMBL8226 0.91 ABL1 (1.00) ABL1SRCPKMYT1BCREPHB6
Dasatinib Anhydrous SCHEMBL29381185 0.91 ABL1 (1.00) ABL1SRCPKMYT1BCREPHB6
Dasatinib Anhydrous SCHEMBL28350326 0.91 ABL1 (1.00) ABL1SRCPKMYT1BCREPHB6
Dasatinib Anhydrous SCHEMBL1705152 0.90 ABL1 (0.98) ABL1SRCPKMYT1BCREPHB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019173224-A1 DEUTERATED COMPOUNDS AND CHIMERAS AND USES THEREOF BIOTHERYX, INC. (US) 2019-09-12 WO disclosed
US-20110212475-A1 Fluorescently Or Spin-Labeled Kinases For Rapid Screening And Identification Of Novel Kinase Inhibitor Scaffolds MAX-PLANCK GESELLSCHAFT ZUR FORDERUNG DER WISSENSCHAFTEN E.V. (DE) 2011-09-01 US disclosed