SCHEMBL12299265

SCHEMBL12299265

CN(CO)/C(N)=N\C1(C)CC(c2ccccc2)Oc2ccc(Br)cc21

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 3/20 0.37
BACE1 P56817 6/20 0.33
KCNH2 Q12809 1/20 0.33
ALOX12 P18054 1/20 0.32
KDM1A O60341 3/20 0.32
RCOR1 Q9UKL0 3/20 0.32
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12300142 0.88 AKR1B1 (0.36) AKR1B1ALOX12AR
SCHEMBL12299283 0.87 AKR1B1 (0.36) AKR1B1BACE1KCNH2ALOX12AR
SCHEMBL12299271 0.86 AKR1B1 (0.33) AKR1B1BACE1
SCHEMBL12299015 0.73 AKR1B1 (0.32) AKR1B1BACE1
SCHEMBL14053922 0.70 AKR1B1 (0.43) AKR1B1BACE1KCNH2KDM1ARCOR1
SCHEMBL14053664 0.70 AKR1B1 (0.43) AKR1B1BACE1KCNH2KDM1ARCOR1
SCHEMBL16136524 0.67 AKR1B1 (0.38) AKR1B1BACE1AR
SCHEMBL27278870 0.67 AKR1B1 (0.75) AKR1B1
SCHEMBL12246365 0.67 AKR1B1 (0.46) AKR1B1AR
SCHEMBL1822169 0.66 AKR1B1 (0.44) AKR1B1BACE1KCNH2ALOX12AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110218192-A1 Inhibitors Of Beta-Secretase VITAE PHARMACEUTICALS, INC. (US) 2011-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110218192-A1 Inhibitors Of Beta-Secretase BACE1, BACE2, APP AKR1B1 2656/4885BACE1 1/4885KCNH2 2890/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.