SCHEMBL12331981

SCHEMBL12331981

Cc1cccnc1N1CCN(C(=O)NCCc2ccccc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 2/20 0.57
TRPV1 Q8NER1 4/20 0.56
TSHR P16473 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CHRM4 P08173 2/20 0.54
KIT P10721 1/20 0.52
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPK1 P28482 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PARP1 P09874 1/20 0.49
TGM2 P21980 1/20 0.49
SMO Q99835 1/20 0.48
TPSAB1 Q15661 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13930757 0.86 CHRM4 (0.70) P2RY12TRPV1TSHRHSD17B10CHRM4
SCHEMBL13930741 0.86 CHRM4 (0.56) P2RY12TSHRHSD17B10CHRM4KIT
SCHEMBL13548403 0.86 P2RY12 (0.55) P2RY12TSHRHSD17B10CHRM4KIT
SCHEMBL12190509 0.84 TSHR (0.53) P2RY12TSHRHSD17B10CHRM4KIT
SCHEMBL12214313 0.84 KDM4E (0.58) P2RY12TSHRHSD17B10CHRM4KIT
SCHEMBL12190505 0.84 GAA (0.64) TRPV1HSD17B10CHRM4
SCHEMBL31298090 0.83 KDM4E (0.66) P2RY12HSD17B10CHRM4KITKDM4E
SCHEMBL12190517 0.83 GRM5 (0.58) P2RY12TSHRHSD17B10CHRM4KIT
SCHEMBL13377920 0.81 CHRM4 (0.59) P2RY12TRPV1CHRM4
SCHEMBL14423759 0.79 P2RY12 (0.59) P2RY12TRPV1CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942106-B1 Therapeutic agents useful for treating pain EURO CELTIQUE SA (LU) 2011-09-14 EP disclosed