SCHEMBL12333147

SCHEMBL12333147

COC(=O)NC(C(=O)N1C[C@@H](C)C[C@H]1c1nc2cc(I)ccc2[nH]1)C(C)C

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.55
KCNH2 Q12809 1/20 0.55
CYP3A4 P08684 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12333040 1.00 CYP2C9 (0.55) CYP2C9KCNH2CYP3A4
SCHEMBL1914105 1.00 CYP2C9 (0.55) CYP2C9KCNH2CYP3A4
SCHEMBL14655351 0.91 CYP2C9 (0.46) CYP2C9KCNH2CYP3A4
SCHEMBL14841664 0.91 CYP2C9 (0.46) CYP2C9KCNH2CYP3A4
SCHEMBL14655274 0.91 CYP2C9 (0.46) CYP2C9KCNH2CYP3A4
SCHEMBL12509506 0.90 CYP2C9 (0.60) CYP2C9KCNH2CYP3A4
SCHEMBL15045762 0.89 CYP2C9 (0.55) CYP2C9KCNH2CYP3A4
SCHEMBL12423487 0.89 CYP2C9 (0.58) CYP2C9KCNH2CYP3A4
SCHEMBL15984499 0.89 CYP2C9 (0.55) CYP2C9KCNH2CYP3A4
SCHEMBL15048011 0.88 CYP2C9 (0.45) CYP2C9KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011119853-A1 ANALOGUES FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-09-29 WO disclosed