SCHEMBL12336804

SCHEMBL12336804

O=CC(c1c2c(nn1-c1ccc(Cl)cc1)CCC2)C1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.53
PTGS2 P35354 5/20 0.38
SRC P12931 3/20 0.36
ENPP2 Q13822 1/20 0.36
GABRA1 P14867 3/20 0.36
GABRA2 P47869 3/20 0.36
CNR1 P21554 2/20 0.34
CNR2 P34972 2/20 0.34
PTGS1 P23219 3/20 0.34
ADORA3 P0DMS8 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1712493 0.98 NR1H4 (0.51) NR1H4PTGS2SRCENPP2GABRA1
SCHEMBL2381928 0.81 NR1H4 (0.59) NR1H4PTGS2SRCENPP2GABRA1
SCHEMBL1712723 0.80 NR1H4 (0.53) NR1H4PTGS2ENPP2GABRA1GABRA2
SCHEMBL2382733 0.80 NR1H4 (0.62) NR1H4PTGS2SRCENPP2GABRA1
SCHEMBL1712067 0.79 NR1H4 (0.54) NR1H4PTGS2ENPP2GABRA1GABRA2
SCHEMBL2383338 0.79 NR1H4 (0.54) NR1H4PTGS2ENPP2GABRA1GABRA2
SCHEMBL2381422 0.79 NR1H4 (0.57) NR1H4PTGS2ENPP2GABRA1GABRA2
SCHEMBL1712371 0.79 NR1H4 (0.57) NR1H4PTGS2ENPP2GABRA1GABRA2
SCHEMBL1712621 0.79 NR1H4 (0.55) NR1H4PTGS2ENPP2CNR1CNR2
SCHEMBL1712617 0.79 NR1H4 (0.55) NR1H4PTGS2ENPP2CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011117163-A1 CYCLOPENTYL - AND CYCLOHEPTYLPYRAZOLES AS FXR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2011-09-29 WO disclosed