SCHEMBL12371159

SCHEMBL12371159

C=CC(=O)Nc1cccc(Sc2nc(Nc3cc(C)c(C4CCN(C)CC4)cc3C)nc3ccnn23)c1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.43
JAK3 P52333 7/20 0.39
BTK Q06187 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12396278 0.93 EGFR (0.48) EGFRJAK3BTK
SCHEMBL12371157 0.90 EGFR (0.43) EGFRJAK3BTK
SCHEMBL12371164 0.85 EGFR (0.40) EGFRJAK3BTK
SCHEMBL12396288 0.85 EGFR (0.45) EGFRJAK3BTK
SCHEMBL12371153 0.84 EGFR (0.46) EGFRJAK3BTK
SCHEMBL12371144 0.84 EGFR (0.56) EGFRJAK3BTK
SCHEMBL12371138 0.83 EGFR (0.43) EGFRJAK3BTK
SCHEMBL12397315 0.80 EGFR (0.61) EGFRJAK3BTK
SCHEMBL12396330 0.79 EGFR (0.48) EGFRBTK
SCHEMBL12398401 0.79 EGFR (0.49) EGFRJAK3BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9879028-B2 Compounds that modulate EGFR activity and methods for treating or preventing conditions therewith Gatekeeper Pharmaceuticals, Inc. (US) 2018-01-30 US disclosed
US-20140011810-A1 Compounds that Modulate EGFR Activity and Methods for Treating or Preventing Conditions Therewith Gatekeeper Pharmaceuticals, Inc. (US) 2014-01-09 US disclosed
US-20110207736-A1 COMPOUNDS THAT MODULATE EGFR ACTIVITY AND METHODS FOR TREATING OR PREVENTING CONDITIONS THEREWITH Gatekeeper Pharmaceuticals, Inc. 2011-08-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110207736-A1 COMPOUNDS THAT MODULATE EGFR ACTIVITY AND METHODS FOR TREATING OR PREVENTING CONDITIONS THEREWITH EGFR, ERBB2, BRCA1 EGFR 1/4885JAK3 254/4885BTK 147/4885
US-20140011810-A1 Compounds that Modulate EGFR Activity and Methods for Treating or Preventing Conditions Therewith EGFR, ERBB2, BRCA1 EGFR 1/4885JAK3 254/4885BTK 147/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.