SCHEMBL12396015

SCHEMBL12396015

Cc1ccc(C(=O)Nc2cc(-c3cccc(F)c3)sc2C(=O)O)cc1

nearest known ligand 0.82

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.73
MEN1 O00255 3/20 0.73
KMT2A Q03164 3/20 0.73
MAPT P10636 1/20 0.73
CRHBP P24387 1/20 0.73
CRHR2 Q13324 1/20 0.73
KDM4E B2RXH2 1/20 0.62
HPGD P15428 2/20 0.56
P2RY14 Q15391 1/20 0.54
PTPN1 P18031 4/20 0.52
PTPRF P10586 1/20 0.52
ALDH1A1 P00352 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2157985 0.91 POLB (0.67) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL12396010 0.90 MEN1 (0.60) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL12396019 0.83 PTPN1 (0.64) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL12396017 0.82 MEN1 (0.54) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL12396099 0.82 DYRK1A (0.54) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL12396020 0.81 KDM4E (0.53) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL3075700 0.81 POLB (0.71) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL16303152 0.80 POLB (0.72) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL2157766 0.78 MAPT (0.67) POLBMEN1KMT2AMAPTCRHBP
SCHEMBL14048862 0.77 POLB (0.59) POLBMEN1KMT2AMAPTCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7985769-B2 Compounds and methods for the treatment or prevention of Flavivirus infections VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-26 US disclosed
US-7985769-B2 Compounds and methods for the treatment or prevention of Flavivirus infections VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-07-26 US disclosed
EP-2206709-A2 Thiophene derivatives as antiviral agents for flavivirus infection Virochem Pharma Inc. (CA) 2010-07-14 EP disclosed