SCHEMBL1240328

SCHEMBL1240328

CC(C(=O)O)(c1cccc(Br)c1)N1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 7/20 0.47
HPGD P15428 1/20 0.44
ALDH1A1 P00352 4/20 0.43
GLA P06280 1/20 0.43
CYP2B6 P20813 1/20 0.42
CHRNA1 P02708 1/20 0.42
CHRNG P07510 1/20 0.42
CHRNB1 P11230 1/20 0.42
CHRNB2 P17787 1/20 0.42
SLC6A2 P23975 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CHRND Q07001 1/20 0.42
GAA P10253 2/20 0.41
TP53 P04637 1/20 0.40
KDM4E B2RXH2 2/20 0.39
POLB P06746 1/20 0.39
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7592805 0.82 CHRM3 (0.57) CHRM3CYP2B6GAASMN1; SMN2
SCHEMBL2126740 0.81 CYP2B6 (0.59) CHRM3CYP2B6
SCHEMBL3043721 0.81 CYP2B6 (0.59) CHRM3CYP2B6
SCHEMBL4444477 0.81 CYP2B6 (0.59) CHRM3CYP2B6
SCHEMBL2127676 0.81 CYP2B6 (0.59) CHRM3CYP2B6
SCHEMBL19690280 0.78 CYP2B6 (0.59) CHRM3HPGDALDH1A1GLACYP2B6
SCHEMBL13653551 0.76 CYP2B6 (0.62) CHRM3HPGDALDH1A1GLACYP2B6
SCHEMBL15123482 0.74 KMT2A (0.45) ALDH1A1GAAMEN1KMT2ASMN1; SMN2
SCHEMBL18982762 0.74 KMT2A (0.45) ALDH1A1GAAMEN1KMT2ASMN1; SMN2
SCHEMBL826639 0.74 KMT2A (0.45) ALDH1A1GAAMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879839-B2 For treatment and prevention of cardiac arrhythmias; (+-)-2-Morpholin-4-yl-2-phenyl-1,1-dipyridin-3-yl-ethanol; (+-)-2-[(2-methoxyethyl)(methyl)amino]-2-phenyl-1,1-dipyridin-3-ylethanol MERCK SHARP & DOHME CORP. (US) 2011-02-01 US disclosed