SCHEMBL12409247

SCHEMBL12409247

COc1ccc(-c2cnc3c(NCc4cnccn4)nccn23)cc1OC

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FYN P06241 5/20 0.45
ADORA3 P0DMS8 1/20 0.45
TTK P33981 10/20 0.43
PAX8 Q06710 1/20 0.41
SRC P12931 1/20 0.41
ATP1A1 P05023 1/20 0.39
ATP1B1 P05026 1/20 0.39
ATP1A3 P13637 1/20 0.39
ATP1B2 P14415 1/20 0.39
ATP1A2 P50993 1/20 0.39
ATP1B3 P54709 1/20 0.39
FXYD2 P54710 1/20 0.39
ATP1A4 Q13733 1/20 0.39
PDE10A Q9Y233 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12409234 0.85 FYN (0.54) FYNADORA3TTK
SCHEMBL12409242 0.84 TTK (0.56) FYNADORA3TTKPAX8ATP1A1
SCHEMBL12409314 0.82 MAPK1 (0.50) FYNTTK
SCHEMBL12409298 0.82 MAPK1 (0.48) FYNADORA3TTKPDE10A
SCHEMBL2178662 0.82 TTK (0.48) FYNADORA3TTKPDE10A
SCHEMBL3470277 0.81 FYN (0.54) FYNTTK
SCHEMBL12409308 0.80 FYN (0.59) FYNADORA3TTK
SCHEMBL12409292 0.80 FYN (0.60) FYNTTK
SCHEMBL12409321 0.80 FYN (0.48) FYNTTKATP1A1ATP1B1ATP1A3
SCHEMBL12409252 0.79 ZAP70 (0.48) FYNTTKPAX8PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS CYP3A5, HAVCR2, CYP3A43 FYN 3511/4885ADORA3 4222/4885TTK 3239/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.