SCHEMBL12425243

SCHEMBL12425243

Bc1cnc(Cl)nc1NC1CCCCCC1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.68
AXL P30530 1/20 0.54
MEN1 O00255 1/20 0.41
PDE4A P27815 1/20 0.41
KDM4E B2RXH2 2/20 0.40
GAA P10253 1/20 0.40
ADORA3 P0DMS8 8/20 0.39
ADORA1 P30542 7/20 0.39
ADORA2A P29274 5/20 0.39
HPGDS O60760 1/20 0.39
PDE10A Q9Y233 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13812811 0.98 KMT2A (0.65) KMT2AAXLMEN1PDE4AKDM4E
SCHEMBL17179514 0.84 KMT2A (0.49) KMT2AAXLADORA3ADORA1ADORA2A
SCHEMBL16438333 0.84 KMT2A (0.49) KMT2AAXLADORA3ADORA1ADORA2A
SCHEMBL13768978 0.84 MAPK1 (0.50) KMT2AAXLADORA3
SCHEMBL1937546 0.83 KMT2A (0.71) KMT2AAXLMEN1PDE4AKDM4E
SCHEMBL1934159 0.81 KMT2A (0.69) KMT2AAXLMEN1PDE4AKDM4E
SCHEMBL24799800 0.81 KMT2A (0.68) KMT2AAXLMEN1PDE4AKDM4E
SCHEMBL2302601 0.81 KMT2A (0.68) KMT2AAXLMEN1PDE4AKDM4E
SCHEMBL19244047 0.81 KMT2A (0.68) KMT2AAXLMEN1PDE4AKDM4E
SCHEMBL21593571 0.81 KMT2A (0.68) KMT2AAXLMEN1PDE4APDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101409-A1 PYRROLOPYRIMIDINE COMPOUNDS AS INHIBITORS OF CDK4/6 NOVARTIS AG (CH) 2011-08-25 WO disclosed