SCHEMBL12426730

SCHEMBL12426730

O=C(O)CC(c1cccnc1)c1ccc2[nH]nc(Cl)c2c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.44
CTSA P10619 6/20 0.41
SUCNR1 Q9BXA5 2/20 0.39
FFAR1 O14842 1/20 0.39
TBXAS1 P24557 1/20 0.39
PHGDH O43175 1/20 0.39
DYRK1A Q13627 3/20 0.38
CDK7 P50613 1/20 0.38
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
ITGA2B P08514 1/20 0.36
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2303540 0.88 KCNA5 (0.43) PDE4DDYRK1ACDK7ITGB3ITGAV
SCHEMBL14495207 0.88 MAPK1 (0.40) CTSAFFAR1KEAP1MAPK1
SCHEMBL14495206 0.88 MAPK1 (0.40) CTSAFFAR1KEAP1MAPK1
SCHEMBL13157460 0.87 PDE4D (0.44) PDE4DDYRK1ACDK7MAPK1
SCHEMBL27742058 0.85 MAP2K4 (0.38) PDE4DDYRK1ACDK7
SCHEMBL2302724 0.80 SLC6A2 (0.44) DYRK1A
SCHEMBL2301515 0.76 ATM (0.42) MAPK1
SCHEMBL14495196 0.76 FFAR1 (0.40) CTSAFFAR1KEAP1NFE2L2MAPK1
SCHEMBL13157447 0.76 MAPK1 (0.39) MAPK1
SCHEMBL13157449 0.76 MAPK1 (0.39) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2351737-A1 3-Amino-1-arylpropyl indoles and aza-substituted indoles F. Hoffmann-La Roche AG (CH) 2011-08-03 EP disclosed
WO-2007062996-A1 3-AMINO-1-ARYLPROPYL INDOLES AND AZA-SUBSTITUTED INDOLES F. HOFFMANN-LA ROCHE AG (CH) 2007-06-07 WO disclosed