SCHEMBL12433712

SCHEMBL12433712

CCCN1C(=O)[C@@H](N)CCc2ccccc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
DRD4 P21917 6/20 0.44
CHRM2 P08172 5/20 0.44
CHRM4 P08173 5/20 0.44
CHRM5 P08912 5/20 0.44
CHRM1 P11229 5/20 0.44
DRD2 P14416 5/20 0.44
CHRM3 P20309 5/20 0.44
DRD3 P35462 5/20 0.44
MTNR1A P48039 1/20 0.44
ADRB2 P07550 1/20 0.44
ADRB1 P08588 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
ACE P12821 2/20 0.43
ANPEP P15144 3/20 0.43
ALDH1A1 P00352 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14005648 0.88 DRD4 (0.51) DRD4CHRM2CHRM4CHRM5CHRM1
SCHEMBL7347045 0.82 ACE (0.56) ACEMEN1KMT2AXIAP
SCHEMBL12893387 0.81 ACE (0.48) ACE
SCHEMBL4992795 0.80 ANPEP (0.49) DRD4DRD2ANPEP
SCHEMBL2276278 0.80 ANPEP (0.49) DRD4DRD2ANPEP
SCHEMBL5638597 0.80 ANPEP (0.49) DRD4DRD2ANPEP
SCHEMBL13899160 0.80 ACE (0.51) MTNR1AACEXIAP
Hydrochloric Acid SCHEMBL2279099 0.79 ANPEP (0.50) DRD4DRD2ANPEP
SCHEMBL5014806 0.79 ANPEP (0.42) ANPEPALDH1A1HTR2A
SCHEMBL199165 0.79 PDPK1 (0.59) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989441-B2 Organic compounds NOVARTIS AG (CH) 2011-08-02 US disclosed