SCHEMBL12436385

SCHEMBL12436385

CC(C)(C)OC(=O)N1C(c2nc(-c3ccc(-c4ccc(-c5c[nH]c(C6[C@H]7CC[C@H](C7)N6C(=O)OC(C)(C)C)n5)cc4)cc3)c[nH]2)[C@H]2CC[C@@H]1C2

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PREP P48147 3/20 0.42
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
KAT2B Q92831 1/20 0.37
HSD11B1 P28845 1/20 0.37
GPR119 Q8TDV5 5/20 0.37
JAK1 P23458 2/20 0.36
HTT P42858 1/20 0.35
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPN6 P29350 1/20 0.35
SCN9A Q15858 1/20 0.35
SCN3A Q9NY46 1/20 0.35
SCN5A Q14524 1/20 0.35
KCNK3 O14649 3/20 0.34
KCNK9 Q9NPC2 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17066303 1.00 PREP (0.42) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL889338 0.94 KCNK3 (0.41) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL12436928 0.94 PREP (0.41) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL12436556 0.94 PREP (0.41) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL16062559 0.94 KCNK3 (0.41) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL18426928 0.94 KCNK3 (0.41) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL12436927 0.92 PREP (0.41) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL16062569 0.90 PREP (0.40) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL16020769 0.90 PREP (0.37) PREPCHRM2CHRM1CHRM3KAT2B
SCHEMBL16020770 0.90 PREP (0.37) PREPCHRM2CHRM1CHRM3KAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091532-A1 HEPATITIS C INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-04 WO disclosed