SCHEMBL12440536

SCHEMBL12440536

Clc1ccc(-c2ccc(CCc3ccc(CN4CCCC4)cc3)nc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
MCHR1 Q99705 9/20 0.54
CHRM1 P11229 5/20 0.53
HTR2A P28223 5/20 0.53
HRH3 Q9Y5N1 3/20 0.53
HRH4 Q9H3N8 1/20 0.53
LSS P48449 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C19 P33261 1/20 0.49
CHEK1 O14757 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12441452 0.99 KDM4E (0.58) KDM4EALDH1A1MCHR1CHRM1HTR2A
SCHEMBL12440426 0.88 HRH3 (0.57) KDM4EALDH1A1MCHR1HRH3LSS
SCHEMBL12440554 0.87 CHKA (0.47) KDM4EALDH1A1MCHR1CHRM1HTR2A
SCHEMBL12440425 0.85 MCHR1 (0.58) KDM4EALDH1A1MCHR1CHRM1HTR2A
SCHEMBL12440218 0.85 MCHR1 (0.45) KDM4EALDH1A1MCHR1CHRM1HTR2A
SCHEMBL12441461 0.85 MCHR1 (0.57) MCHR1CHRM1HTR2AHRH3HRH4
SCHEMBL12440662 0.83 HRH3 (0.57) KDM4EALDH1A1MCHR1CHRM1HTR2A
SCHEMBL12441111 0.82 LSS (0.41) MCHR1CHRM1HTR2AHRH3LSS
SCHEMBL12440034 0.82 KDM4E (0.60) KDM4EALDH1A1MCHR1CHRM1HTR2A
SCHEMBL12441459 0.80 MCHR1 (0.70) KDM4EALDH1A1MCHR1CHRM1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed