SCHEMBL12440742

SCHEMBL12440742

CC1CCN(C2CCCC(c3ccc(-c4ccc(-c5ccc(Cl)cc5)cn4)cc3)C2)CC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.42
MAOB P27338 1/20 0.42
CHRM1 P11229 2/20 0.37
HTR2A P28223 2/20 0.37
MCHR1 Q99705 2/20 0.37
HSD11B1 P28845 1/20 0.36
CNR2 P34972 1/20 0.36
HRH3 Q9Y5N1 7/20 0.35
PROKR1 Q8TCW9 1/20 0.35
SLC18A3 Q16572 1/20 0.34
MITF O75030 1/20 0.34
RAB9A P51151 1/20 0.34
DGAT1 O75907 1/20 0.34
KCNH2 Q12809 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
PRCP P42785 1/20 0.33
KDM2B Q8NHM5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440216 0.94 KDM1A (0.43) KDM1AMAOBCHRM1HTR2AMCHR1
SCHEMBL5227157 0.84 MCHR1 (0.57) CHRM1HTR2AMCHR1
SCHEMBL5226871 0.78 MCHR1 (0.59) CHRM1HTR2AMCHR1HRH3
SCHEMBL12441406 0.75 MAOB (0.39) KDM1AMAOBCHRM1HTR2AMCHR1
SCHEMBL12440550 0.74 MAOB (0.40) KDM1AMAOBCHRM1HTR2AMCHR1
SCHEMBL5226268 0.74 MCHR1 (0.50) CHRM1HTR2AMCHR1HRH3KCNH2
SCHEMBL12440597 0.73 CNR2 (0.49) MCHR1CNR2DGAT1KCNH2
SCHEMBL18936735 0.72 ESR2 (0.51) HRH3SLC18A3
SCHEMBL12441099 0.68 MCHR1 (0.72) CHRM1HTR2AMCHR1HRH3
SCHEMBL18790890 0.68 NPC1 (0.45) KDM1ARAB9ADGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed