SCHEMBL1245862

SCHEMBL1245862

CC(=O)C1=C(C)N(c2cccc(C(F)(F)F)c2)C(=O)N(CCNC(=O)O)C1c1ccc(C#N)cc1

nearest known ligand 0.80

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.80
CYP2C9 P11712 4/20 0.80
CYP3A4 P08684 4/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13872684 0.92 ELANE (0.77) ELANECYP2C9CYP3A4
SCHEMBL8288689 0.90 ELANE (0.70) ELANECYP2C9CYP3A4
SCHEMBL13872736 0.90 ELANE (0.81) ELANECYP2C9CYP3A4
SCHEMBL13872728 0.89 ELANE (0.85) ELANECYP2C9CYP3A4
SCHEMBL13872730 0.89 ELANE (0.85) ELANECYP2C9CYP3A4
SCHEMBL1245224 0.89 ELANE (1.00) ELANECYP2C9CYP3A4
SCHEMBL3482543 0.89 ELANE (1.00) ELANECYP2C9CYP3A4
SCHEMBL5095677 0.88 ELANE (0.82) ELANECYP2C9CYP3A4
SCHEMBL8287682 0.86 ELANE (0.82) ELANECYP2C9CYP3A4
SCHEMBL3482560 0.86 ELANE (0.85) ELANECYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730121-B1 1,4-DIARYL-DIHYDROPYRIMIDIN-2-ONES AND THEIR USE AS HUMAN NEUTROPHIL ELASTASE INHIBITORS BAYER IP GMBH (DE) 2013-08-07 EP disclosed
US-7893073-B2 Heterocyclic derivatives BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-02-22 US disclosed