SCHEMBL12460899

SCHEMBL12460899

CC(=O)c1c([C@@H]2C[C@H]3CC[C@@H](C2)N3C(=O)C(C)(CO)CO)nc2c(-c3ccc(-c4ccc(O)c(F)c4)nc3)cnn2c1N

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTOR P42345 4/20 0.40
RPTOR Q8N122 4/20 0.40
MLST8 Q9BVC4 4/20 0.40
BRAF P15056 2/20 0.32
NPC1 O15118 4/20 0.31
RAB9A P51151 4/20 0.31
KDM4E B2RXH2 3/20 0.31
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C19 P33261 1/20 0.31
RECQL P46063 1/20 0.31
MAP3K12 Q12852 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
MAPT P10636 1/20 0.30
ALK Q9UM73 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14245944 0.91 MTOR (0.39) MTORRPTORMLST8BRAFMAPT
SCHEMBL14245942 0.91 MTOR (0.39) MTORRPTORMLST8BRAFMAPT
SCHEMBL12460267 0.91 MTOR (0.39) MTORRPTORMLST8BRAFMAPT
SCHEMBL14298177 0.91 MTOR (0.39) MTORRPTORMLST8BRAFMAPT
SCHEMBL12460278 0.89 MTOR (0.51) MTORRPTORMLST8NPC1RAB9A
SCHEMBL12460874 0.89 MTOR (0.51) MTORRPTORMLST8NPC1RAB9A
SCHEMBL14245547 0.89 MTOR (0.51) MTORRPTORMLST8NPC1RAB9A
SCHEMBL2147372 0.89 MTOR (0.51) MTORRPTORMLST8NPC1RAB9A
SCHEMBL2147228 0.85 MTOR (0.53) MTORRPTORMLST8BRAF
SCHEMBL14245610 0.85 MTOR (0.53) MTORRPTORMLST8BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011090935-A1 PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-28 WO disclosed